Aladinskaya Anastasia V.
Количество цитирований статей в журналах по данным
Web of Science: 62,
Scopus: 87
IstinaResearcherID (IRID): 21391629
Деятельность
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Статьи в журналах
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2021
Novel potent PSMA ligands and their docetaxel conjugates: in vitro and in vivo evaluation
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Machulkin A.E.,
Uspenskaya A.A.,
Ber A.P.,
Petrov S.A.,
Nimenko E.A.,
Zyk N.U.,
Ivanenkov Y.A.,
Aladinskaya A.V.,
Skvortsov D.A.,
Borisova Y.A.,
Smirnova G.B.,
Pokrovsky V.S.,
Vaneev A.N.,
Erofeev A.S.,
Gorelkin P.V.,
Beloglazkina E.K.,
Zyk N.V.,
Majouga A.G.
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в журнале FEBS open bio, издательство John Wiley & Sons Inc. (United States), том 11, № S1, с. 43-44
DOI
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2021
Synthesis and Biological Evaluation of PSMA Ligands with Aromatic Residues and Fluorescent Conjugates Based on Them
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Machulkin A.E.,
Shafikov R.R.,
Uspenskaya A.A.,
Petrov S.A.,
Ber A.P.,
Skvortsov D.A.,
Nimenko E.A.,
Zyk N.U.,
Smirnova G.B.,
Pokrovsky V.S.,
Abakumov M.A.,
Saltykova I.V.,
Akhmirov R.T.,
Garanina A.S.,
Polshakov V.I.,
Saveliev O.Y.,
Ivanenkov Y.A.,
Aladinskaya A.V.,
Finko A.V.,
Yamansarov E.U.,
Krasnovskaya O.O.,
Erofeev A.S.,
Gorelkin P.V.,
Dontsova O.A.,
Beloglazkina E.K.,
Zyk N.V.,
Khazanova E.S.,
Majouga A.G.
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в журнале Journal of Medicinal Chemistry, издательство American Chemical Society (United States), том 64, № 8, с. 4532-4552
DOI
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2021
Synthesis and biological evaluation of PSMA ligands with aromatic residues and fluorescent conjugates based on them
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Machulkin A.E.,
Shafikov R.R.,
Uspenskaya A.A.,
Petrov S.A.,
Ber A.P.,
Skvortsov D.A.,
Nimenko E.A.,
Zyk N.U.,
Smirnova G.B.,
Pokrovsky V.S.,
Abakumov M.A.,
Saltykova I.V.,
Akhmirov R.T.,
Garanina A.S.,
Polshakov V.I.,
Saveliev O.Y.,
Ivanenkov Y.A.,
Aladinskaya A.V.,
Finko A.V.,
Yamansarov E.U.,
Krasnovskaya O.O.,
Erofeev A.S.,
Gorelkin P.V.,
Dontsova O.A.,
Beloglazkina E.K.,
Zyk N.V.,
Khazanova E.S.,
Majouga A.G.
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в журнале Journal of Medicinal Chemistry, издательство American Chemical Society (United States)
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2020
Identification of pyrrolo-pyridine derivatives as novel class of antibacterials
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Veselov Mark S.,
Ivanenkov Yan A.,
Yamidanov Renat S.,
Osterman Ilya A.,
Sergiev Petr V.,
Aladinskiy Vladimir A.,
Aladinskaya Anastasia V.,
Terentiev Victor A.,
Ayginin Andrey A.,
Skvortsov Dmitry A.,
Komarova Katerina S.,
Chemeris Alexey V.,
Baimiev Alexey Kh,
Sofronova Alina A.,
Machulkin Alexey E.,
Petrov Rostislav A.,
Maklakova Svetlana Yu,
Bezrukov Dmitry S.,
Filkov Gleb I.,
Zainullina Liana F.,
Maximova Marina A.,
Zileeva Zulfiya R.,
Kartsev Victor G.,
Vakhitova Yulia V.,
Dontsova Olga A.
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в журнале Molecular Diversity, издательство Springer Nature (Switzerland), том 24, № 1, с. 233-239
DOI
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2019
2-Pyrazol-1-yl-thiazole derivatives as novel highly potent antibacterials
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Ivanenkov Yan A.,
Yamidanov Renat S.,
Osterman Ilya A.,
Sergiev Petr V.,
Aladinskiy Vladimir A.,
Aladinskaya Anastasia V.,
Terentiev Victor A.,
Veselov Mark S.,
Ayginin Andrey A.,
Skvortsov Dmitry A.,
Komarova Katerina S.,
Sadovnikov Sergey V.,
Rustam Matniyazov,
Sofronova Alina A.,
Malyshev Alexander S.,
Machulkin Alexey E.,
Petrov Rostislav A.,
Dmitrii Lukianov,
Svetlana Iarovenko,
Bezrukov Dmitry S.,
Baymiev Andrey Kh,
Dontsova Olga A.
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в журнале Journal of Antibiotics, издательство Japan Antibiotics Research Association/Nihon Koseibusshitsu Gakujutsu Kyogikai (Japan), том 72, с. 827-833
DOI
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2019
Deep learning enables rapid identification of potent DDR1 kinase inhibitors
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Zhavoronkov Alex,
Ivanenkov Yan A.,
Aliper Alex,
Veselov Mark S.,
Aladinskiy Vladimir A.,
Aladinskaya Anastasiya V.,
Terentiev Victor A.,
Polykovskiy Daniil A.,
Kuznetsov Maksim D.,
Asadulaev Arip,
Volkov Yury,
Zholus Artem,
Shayakhmetov Rim R.,
Zhebrak Alexander,
Minaeva Lidiya I.,
Zagribelnyy Bogdan A.,
Lee Lennart H.,
Soll Richard,
Madge David,
Xing Li,
Guo Tao,
Aspuru-Guzik Alán
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в журнале Nature Biotechnology, издательство Nature Publishing Group (United Kingdom)
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2019
Identification of N-Substituted Triazolo-azetidines as Novel Antibacterials using pDualrep2 HTS Platform
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Ivanenkov Yan A.,
Yamidanov Renat S.,
Osterman Ilya A.,
Sergiev Petr V.,
Aladinskiy Vladimir A.,
Aladinskaya Anastasia V.,
Terentiev Victor A.,
Veselov Mark S.,
Ayginin Andrey A.,
Skvortsov Dmitry A.,
Komarova Katerina S.,
Chemeris Alexey V.,
Baimiev Alexey Kh,
Sofronova Alina A.,
Malyshev Alexander S.,
Machulkin Alexey E.,
Petrov Rostislav A.,
Bezrukov Dmitry S.,
Filkov Gleb I.,
Puchinina Maria M.,
Zainullina Liana F.,
Maximova Marina A.,
Zileeva Zulfiya R.,
Vakhitova Yulia V.,
Dontsova Olga A.
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в журнале Combinatorial Chemistry and High Throughput Screening, издательство Bentham Science Publishers (Netherlands), том 22, № 5, с. 346-354
DOI
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2019
Identification of Novel Antibacterials Using Machine Learning Techniques
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Ivanenkov Yan A.,
Zhavoronkov Alex,
Yamidanov Renat S.,
Osterman Ilya A.,
Sergiev Petr V.,
Aladinskiy Vladimir A.,
Aladinskaya Anastasia V.,
Terentiev Victor A.,
Veselov Mark S.,
Ayginin Andrey A.,
Kartsev Victor G.,
Skvortsov Dmitry A.,
Chemeris Alexey V.,
Baimiev Alexey Kh,
Sofronova Alina A.,
Malyshev Alexander S.,
Filkov Gleb I.,
Bezrukov Dmitry S.,
Zagribelnyy Bogdan A.,
Putin Evgeny O.,
Puchinina Maria M.,
Dontsova Olga A.
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в журнале Frontiers in pharmacology, издательство Frontiers Media] ([Lausanne, Switzerland), том 10, с. e913
DOI
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2019
Substituted Furanocoumarins as Novel Class of Antibacterial Translation Inhibitors
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Ivanenkov Yan A.,
Yamidanov Renat S.,
Osterman Ilya A.,
Sergiev Petr V.,
Ayginin Andrey A.,
Aladinskiy Vladimir A.,
Aladinskaya Anastasia V.,
Terentiev Victor A.,
Veselov Mark S.,
Skvortsov Dmitry A.,
Komarova Katerina S.,
Chemeris Alexey V.,
Zainullina Liana F.,
Maximova Marina A.,
Zileeva Zulfiya R.,
Vakhitova Yulia V.,
Baimiev Alexey Kh,
Sofronova Alina A.,
Machulkin Alexey E.,
Petrov Rostislav A.,
Bezrukov Dmitry S.,
Puchinina Maria M.,
Dmitrii Lukianov A.,
Dontsova Olga A.
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в журнале Combinatorial Chemistry and High Throughput Screening, издательство Bentham Science Publishers (Netherlands), том 22, № 6, с. 400-410
DOI
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2019
Synthesis and Biological Evaluation of Doxorubicin-containing Conjugate targeting PSMA
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Ivanenkov Yan,
Machulkin Alexey,
Garanina Anastasia,
Skvortsov Dmitry,
Uspenskaya Anastasia,
Deyneka Ekaterina,
Alexander Trofimenko,
Beloglazkina Elena,
Zyk Nikolay,
Koteliansky Victor,
Bezrukov Dmitry,
Aladinskaya Anastasia,
Vorobyeva Nataliya,
Puchinina Maria,
Riabykh Grigory,
Sofronova Alina,
Malyshev Alexander,
Majouga Alexander
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в журнале Bioorganic and Medicinal Chemistry Letters, издательство Pergamon Press Ltd. (United Kingdom), том 29, № 10, с. 1246-1255
DOI
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2019
Synthesis and biological evaluation of Doxorubicin-containing conjugate targeting PSMA
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Ivanenkov Yan A.,
Machulkin Alexey E.,
Garanina Anastasia S.,
Skvortsov Dmitry A.,
Uspenskaya Anastasia A.,
Deyneka Ekaterina,
V,
Trofimenko Alexander,
V,
Beloglazkin Elena K.,
Zyk Nikolay,
V,
Koteliansky Victor E.,
Bezruko Dmitry S.,
Aladinskaya Anastasia V.,
Vorobyeva Nataliya S.,
Puchinina Maria M.,
Ryabykh Grigory K.,
Sofronova Alina A.,
Malyshev Alexander S.,
Majouga Alexander G.
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в журнале Bioorganic and Medicinal Chemistry Letters, издательство Pergamon Press Ltd. (United Kingdom), том 29, № 10, с. 1246-1255
DOI
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2019
Synthesis and biological evaluation of PSMA-targeting paclitaxel conjugates
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Machulkin Alexey E.,
Skvortsov Dmitry A.,
Ivanenkov Yan A.,
Ber Anton P.,
Kavalchuk Mikhail V.,
Aladinskaya Anastasia V.,
Uspenskaya Anastasia A.,
Shafikov Radik R.,
Plotnikova Ekaterina A.,
Yakubovskaya Raisa I.,
Nimenko Ekaterina A.,
Zyk Nikolay U.,
Beloglazkina Elena K.,
Zyk Nikolay V.,
Koteliansky Victor E.,
Majouga Alexander G.
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в журнале Bioorganic and Medicinal Chemistry Letters, издательство Pergamon Press Ltd. (United Kingdom), том 29, № 16, с. 2229-2235
DOI
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2018
Synthesis and Biological Evaluation of Novel Mono- and Bivalent ASGP-R-targeted Drug-conjugates
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Petrov Rostislav A.,
Maklakova Svetlana Yu,
Ivanenkov Yan A.,
Petrov Stanislav A.,
Sergeeva Olga V.,
Yamansarov Emil Yu,
Saltykova Irina V.,
Kireev Igor I.,
Alieva Irina B.,
Deyneka Ekaterina V.,
Sofronova Alina A.,
Aladinskaia Anastasiia V.,
Trofimenko Alexandre V.,
Yamidanov Renat S.,
Kovalev Sergey V.,
Kotelianski Victor E.,
Zatsepin Timofey S.,
Beloglazkina Elena K.,
Majouga Alexander G.
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в журнале Bioorganic and Medicinal Chemistry Letters, издательство Pergamon Press Ltd. (United Kingdom), том 28, № 3, с. 382-387
DOI
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2017
Synthesis and Biological Evaluation of Novel Mono- and Bivalent ASGP-R-targeted Drug-conjugates
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Петров Р.А.,
Маклакова С.Ю.,
Иваненков Ю.А.,
Петров С.А.,
Сергеева О.В.,
Ямансаров Е.Ю.,
Салтыкова И.В.,
Киреев И.И.,
Алиева И.Б.,
Дейнека Е.В.,
Софронова А.А.,
Аладинская А.В.,
Трофименко А.В.,
Ямиданов Р.С.,
Ковалев С.В.,
Котельянский В.Е.
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в журнале Bioorganic and Medicinal Chemistry Letters, издательство Pergamon Press Ltd. (United Kingdom)
DOI
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2016
Small-molecule PSMA ligands. Current state, SAR and perspectives
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Machulkin Alexey E.,
Ivanenkov Yan A.,
Aladinskaya Anastasia V.,
Veselov Mark S.,
Aladinskiy Vladimir A.,
Beloglazkina Elena K.,
Koteliansky Victor E.,
Shakhbazyan Artem G.,
Sandulenko Yuri B.,
Majouga Alexander G.
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в журнале Journal of Drug Targeting, издательство Taylor & Francis (United Kingdom), том 24, № 8, с. 679-693
DOI
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Доклады на конференциях
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2021
Novel potent PSMA ligands and their docetaxel conjugates: in vitro and in vivo evaluation
(Устный)
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Авторы:
Machulkin A.E.,
Uspenskaya A.A.,
Ber A.P.,
Petrov S.A.,
Nimenko E.A.,
Zyk N.U.,
Ivanenkov Y.A.,
Aladinskaya A.V.,
Skvortsov D.A.,
Borisova Y.A.,
Smirnova G.B.,
Pokrovsky V.S.,
Vaneev A.N.,
Erofeev A.S.,
Gorelkin P.V.,
Beloglazkina E.K.,
Zyk N.V.,
Majouga A.G.
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The 45th FEBS Congress, Любляна, Словения, 3-8 июля 2021
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Тезисы докладов
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2021
Novel potent PSMA ligands and their docetaxel conjugates: in vitro and in vivo evaluation
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Machulkin A.E.,
Uspenskaya A.A.,
Ber A.P.,
Petrov S.A.,
Nimenko E.A.,
Zyk N.U.,
Ivanenkov Y.A.,
Aladinskaya A.V.,
Skvortsov D.A.,
Borisova Y.A.,
Smirnova G.B.,
Pokrovsky V.S.,
Vaneev A.N.,
Erofeev A.S.,
Gorelkin P.V.,
Beloglazkina E.K.,
Zyk N.V.,
Majouga A.G.
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в сборнике The 45th FEBS Congress, Любляна, Словения, 3-8 июля 2021, тезисы
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Патенты