Antitumor efficacy of Auger electron emitter In-111 delivered by modular nanotransporter into the nuclei of cells with folate receptor overexpressionстатья
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Дата последнего поиска статьи во внешних источниках: 20 декабря 2019 г.
Аннотация:A new modular nanotransporter (MNT) for the delivery of anticancer agents into the nuclei of cells with folate receptor overexpression was created. An effective method for acceding labeling of this MNT with Auger electron emitter In-111 has been developed. A significant therapeutic effect was observed after a single intratumoral injection of the new In-111-labeled MNT to mice grafted with human cervical carcinoma characterized by folate receptor overexpression.