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Journal of Medicinal Chemistryжурнал

Статьи, опубликованные в журнале

• • 2025 Designing Effective Antimicrobial Agents: Structural Insights into the Antibiofilm Activity of Ionic Liquids
  • Tikhomirov Alexey D., Egorova Ksenia S., Ananikov Valentine P.
  • в журнале Journal of Medicinal Chemistry, издательство American Chemical Society (United States), том 68, № 3, с. 2105-2123 DOI
• • 2025 Pivotal Role of the Intracellular Microenvironment in the High Photodynamic Activity of Cationic Phthalocyanines
  • Bunin Dmitry A., Akasov Roman A., Martynov Alexander G., Stepanova Maria P., Monich Svetlana V., Tsivadze Aslan Yu, Gorbunova Yulia G.
  • в журнале Journal of Medicinal Chemistry, издательство American Chemical Society (United States), том 68, № 1, с. 658-673 DOI
• • 2025 Rational Design of a Potent, Selective, and Metabolically Stable CDK9 Inhibitor to Counteract Osimertinib Resistance through Mcl-1 Suppression and Enhanced BRD4 Co-Targeting
  • Wu Tizhi, Huang Jiali, Zhang Xiankang, Ma Feihai, Yu Shijing, Liu Yifang, Xu Yifan, Wu Shiqi, Finko Alexander V., Li Zhiyu, Feng Li, Bian Jinlei
  • в журнале Journal of Medicinal Chemistry, издательство American Chemical Society (United States), том 68, № 4, с. 4929-4950 DOI
• • 2025 Recent Developments in 14–3–3 Stabilizers for Regulating Protein–Protein Interactions: An Update
  • Tian Yucheng, Li Longjing, Wu Liuyi, Xu Qianqian, Li Yaojie, Pan Huawei, Bing Tiejun, Bai Xiumei, Finko A.V., Li Zhiyu, Bian Jinlei
  • в журнале Journal of Medicinal Chemistry, издательство American Chemical Society (United States), том 68, № 3, с. 2124-2146 DOI
• • 2022 Pt(IV) Prodrugs with Non-Steroidal Anti-inflammatory Drugs in the Axial Position
  • Spector Daniil V., Pavlov Kirill G., Akasov Roman A., Vaneev Alexander N., Erofeev Alexander S., Gorelkin Petr V., Nikitina Vita N., Lopatukhina Elena V., Semkina Alevtina S., Vlasova Kseniya Yu, Skvortsov Dmitrii A., Roznyatovsky Vitaly A., Ul’yanovskiy Nikolay V., Pikovskoi Ilya I., Sypalov Sergey A., Garanina Anastasiia S., Vodopyanov Stepan S., Abakumov Maxim A., Volodina Yulia L., Markova Alina A., Petrova Albina S., Mazur Dmitrii M., Sakharov Dmitry A., Zyk Nikolay V., Beloglazkina Elena K., Majouga Alexander G., Krasnovskaya Olga O.
  • в журнале Journal of Medicinal Chemistry, издательство American Chemical Society (United States), том 65, № 12, с. 8227-8244 DOI
• • 2022 Small Amphiphilic Peptides: Activity Against a Broad Range of Drug-Resistant Bacteria and Structural Insight into Membranolytic Properties
  • Lohan Sandeep, Mandal Dindyal, Choi Wonsuk, Konshina Anastasia G., Tiwari Rakesh K., Efremov Roman G., Maslennikov Innokentiy, Parang Keykavous
  • в журнале Journal of Medicinal Chemistry, издательство American Chemical Society (United States), том 65, № 1, с. 665-687 DOI
• • 2021 HIV-1 gp120 Antagonists Also Inhibit HIV-1 Reverse Transcriptase by Bridging the NNRTI and NRTI Sites
  • Losada Natalie, Ruiz Francesc X., Curreli Francesca, Gruber Kevin, Pilch Alyssa, Altieri Andrea, Kurkin Alexander V., Das Kalyan, Debnath Asim K., Arnold Eddy
  • в журнале Journal of Medicinal Chemistry, издательство American Chemical Society (United States), том 64, № 22, с. 16530-16540 DOI
• • 2021 Mechanisms of the Antiproliferative and Antitumor Activity of Novel Telomerase-Carbonic Anhydrase Dual-Hybrid Inhibitors
  • Plyasova AA, Berrino E., Khan II, Veselovsky AV, Pokrovsky VS, Angeli A., Ferraroni M., Supuran CT, Pokrovskaya MV, Alexandrova SS, Gladilina YA, Sokolov NN, Hilal A., Carta F., Zhdanov DD
  • в журнале Journal of Medicinal Chemistry, издательство American Chemical Society (United States), том 64, № 15 DOI
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  • 2021 Synthesis and Biological Evaluation of PSMA Ligands with Aromatic Residues and Fluorescent Conjugates Based on Them
  • Machulkin A.E., Shafikov R.R., Uspenskaya A.A., Petrov S.A., Ber A.P., Skvortsov D.A., Nimenko E.A., Zyk N.U., Smirnova G.B., Pokrovsky V.S., Abakumov M.A., Saltykova I.V., Akhmirov R.T., Garanina A.S., Polshakov V.I., Saveliev O.Y., Ivanenkov Y.A., Aladinskaya A.V., Finko A.V., Yamansarov E.U., Krasnovskaya O.O., Erofeev A.S., Gorelkin P.V., Dontsova O.A., Beloglazkina E.K., Zyk N.V., Khazanova E.S., Majouga A.G.
  • в журнале Journal of Medicinal Chemistry, издательство American Chemical Society (United States), том 64, № 8, с. 4532-4552 DOI
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  • 2021 Synthesis, characterization and preclinical evaluation of small-molecule prostate-specific membrane antigen targeted monomethyl auristatin E conjugate
  • Machulkin Aleksei E., Uspenskaya Anastasia A., Zyk Nikolay U., Nimenko Ekaterina A., Ber Anton P., Petrov Stanislav A., Polshakov Vladimir I., Shafikov Radik R., Skvortsov Dmitry A., Plotnikova Ekaterina A., Pankratov Andrei A., Smirnova Galina B., Borisova Yulia A., Pokrovsky Vadim S., Kolmogorov Vasilii S., Vaneev Alexander N., Khudyakov A.D., Chepikova Olga E., Kovalev Sergei V., Zamyatnin Andrey A., Erofeev Alexander S., Gorelkin Petr V., Beloglazkina Elena K., Zyk Nikolay V., Khazanova Elena S., Majouga Alexander G.
  • в журнале Journal of Medicinal Chemistry, издательство American Chemical Society (United States), том 64, № 23, с. 17123-17145 DOI
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  • 2020 Acylated 1H-1,2,4-Triazol-5-amines Targeting Human Coagulation Factor XIIa and Thrombin: Conventional and Microscale Synthesis, Anticoagulant Properties, and Mechanism of Action
  • Korff Marvin, Imberg Lukas, Will Jonas M., Bückreiß Nico, Kalinina Svetlana A., Wenzel Benjamin M., Kastner Gregor A., Daniliuc Constantin G., Barth Maximilian, Ovsepyan Ruzanna A., Butov Kirill R., Humpf Hans-Ulrich, Lehr Matthias, Panteleev Mikhail A., Poso Antti, Karst Uwe, Steinmetzer Torsten, Bendas Gerd, Kalinin Dmitrii V.
  • в журнале Journal of Medicinal Chemistry, издательство American Chemical Society (United States) DOI
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  • 2020 Azidothymidine "Clicked" into 1,2,3-Triazoles: First Report on Carbonic Anhydrase-Telomerase Dual-Hybrid Inhibitors
  • Berrino E., Angeli A., Zhdanov D.D., Kiryukhina A.P., Milaneschi A., De_Luca A., Bozdag M., Carradori S., Selleri S., Bartolucci G., Peat T.S., Ferraroni M., Supuran C.T., Carta F.
  • в журнале Journal of Medicinal Chemistry, издательство American Chemical Society (United States), том 63, № 13, с. 7392-7409 DOI
• • 2020 Colchicine Alkaloids and Synthetic Analogues: Current Progress and Perspectives
  • Gracheva Iuliia A., Shchegravina Ekaterina S., Schmalz Hans-Günther, Beletskaya Irina P., Fedorov Alexey Yu
  • в журнале Journal of Medicinal Chemistry, издательство American Chemical Society (United States), том 63, № 19, с. 10618-10651 DOI
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  • 2020 Novel copper-containing cytotoxic agents based on 2-thioxoimidazolones
  • Krasnovskaya Olga, Guk Dmitry A., Naumov Alexey, Nikitina Vita N., Semkina Alevtina, Vlasova Kseniya Yu, Pokrovsky Vadim, Ryabaya Oksana O., Karshieva Saida, Skvortsov Dmitry A., Zhirkina Irina, Shafikov Radik R., Gorelkin Petr, Vaneev Alexander, Erofeev Alexander, Mazur Dmitrii, Tafeenko Viktor Aleksandrovich, Pergushov Vladimir I., Melnikov Mikhail, Soldatov Mikhail A., Shapovalov Victor V., Soldatov Alexander V., Akasov Roman, Gerasimov Vasily, Sakharov Dmitry A., Moiseeva Anna A., Zyk Nikolay Vasil'evich, Beloglazkina Elena K., Majouga Alexander G.
  • в журнале Journal of Medicinal Chemistry, издательство American Chemical Society (United States), том 63, № 21, с. 13031-13063 DOI
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  • 2020 Preclinical Optimization of gp120 Entry Antagonists as anti-HIV-1 Agents with Improved Cytotoxicity and ADME Properties through Rational Design, Synthesis, and Antiviral Evaluation
  • Curreli F., Shahad A., Benedict Victor S.M., Iusupov I.R., Belov D.S., Markov P.O., Kurkin A.V., Altieri A., Debnath A.K.
  • в журнале Journal of Medicinal Chemistry, издательство American Chemical Society (United States), том 63, № 4, с. 1724-1749 DOI
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  • 2019 Are we Opening the Door to a New Era of Medicinal Chemistry or Being Collapsed to a Chemical Singularity?
  • Ivanenkov Yan A., Zagribelnyy Bogdan, Aladinskiy Vladimir
  • в журнале Journal of Medicinal Chemistry, издательство American Chemical Society (United States), том 62, № 22, с. 10026-10043 DOI
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  • 2019 New Rigid Nicotine Analogues, Carrying a Norbornane Moiety, Are Potent Agonists of $\upalpha$7 and $\upalpha$3\ast Nicotinic Receptors
  • Manetti Dina, Garifulina Alexandra, Bartolucci Gianluca, Bazzicalupi Carla, Bellucci Cristina, Chiaramonte Niccolò, Dei Silvia, Mannelli Lorenzo Di Cesare, Ghelardini Carla, Gratteri Paola, Spirova Ekaterina, Shelukhina Irina, Teodori Elisabetta, Varani Katia, Tsetlin Victor, Romanelli Maria Novella
  • в журнале Journal of Medicinal Chemistry, издательство American Chemical Society (United States), том 62, № 4, с. 1887-1901 DOI
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  • 2019 Unforeseen Possibilities To Investigate the Regulation of Polyamine Metabolism Revealed by Novel C-Methylated Spermine Derivatives
  • Khomutov M., Hyvönen M.T., Simonian A., Formanovsky A.A., Mikhura I.V., Chizhov A.O., Kochetkov S.N., Alhonen L., Vepsäläinen J., Keinänen T.A., Khomutov A.R.
  • в журнале Journal of Medicinal Chemistry, издательство American Chemical Society (United States), том 62, № 24, с. 11335-11347
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  • 2019 Water-Soluble Chlorin/Arylaminoquinazoline Conjugate for Photodynamic and Targeted Therapy
  • Otvagin Vasilii F., Kuzmina Natalia S., Krylova Lubov V., Volovetsky Arthur B., Nyuchev Alexander V., Gavryushin Andrei E., Meshkov Ivan N., Gorbunova Yulia G., Romanenko Yuliya V., Koifman Oscar I., Balalaeva Irina V., Fedorov Alexey Yu
  • в журнале Journal of Medicinal Chemistry, издательство American Chemical Society (United States), том 62, № 24, с. 11182-11193 DOI
• • 2017 Discovery of a Novel Series of Tankyrase Inhibitors by a Hybridization Approach
  • Upendra Rao Anumala, Waaler Jo, Yves Nkizinkiko, Alexander Ignatev, Katina Lazarow, Peter Lindemann, Petter Angell Olsen, Sudarshan Murthy, Ezeogo Obaji, Majouga Alexander G., Sergey Leonov, von Kries Jens Peter, Lari Lehtiö, Stefan Krauss, Marc Nazaré
  • в журнале Journal of Medicinal Chemistry, издательство American Chemical Society (United States)
• • 2017 RNA G-quadruplexes in Kirsten ras (KRAS) oncogene as targets for small molecules inhibiting translation
  • Giulia Miglietta, Susanna Cogoi, Jessica Marinello, Giovanni Capranico, Tikhomirov Alexander S., Shchekotikhin Andrey E., and Luigi E.Xodo
  • в журнале Journal of Medicinal Chemistry, издательство American Chemical Society (United States) DOI
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  • 2017 Synthesis and Investigation of Photophysical and Biological Properties of Novel S-Containing Bacteriopurpurinimides
  • Pantushenko Ivan V., Ostroverkhov Petr V., Plotnikova Ekaterina A., Karmakova Tatyana A., Starovoitova Anna V., Burmistrova Nelli V., Yuzhakov Vadim V., Romanko Yuri S., Abakumov Maxim A., Ignatova Anastasiya A., Feofanov Alexey V., Kaplan Mikhail A., Yakubovskaya Raisa I., Tsigankov Anatoliy A., Majouga Alexander G.
  • в журнале Journal of Medicinal Chemistry, издательство American Chemical Society (United States), том 60, № 24, с. 10220-10230 DOI
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  • 2017 Synthesis, antiviral potency, in vitro ADMET and X-ray structure of potent CD4-mimics as entry inhibitors that target the Phe43 cavity of HIV-1 gp120
  • Curreli F., Kwon Y.D., Belov D.S., Ramesh R.R., Kurkin A.V., Altieri A., Kwong P.D., Debnath A.K.
  • в журнале Journal of Medicinal Chemistry, издательство American Chemical Society (United States), том 60, № 7, с. 3124-3153 DOI
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  • 2016 Kinetically Selective Inhibitors of Human Carbonic Anhydrase Isozymes I, II, VII, IX, XII, and XIII
  • Talibov V.O., Linkuviene V., Matulis D., Danielson U.H.
  • в журнале Journal of Medicinal Chemistry, издательство American Chemical Society (United States), том 59, № 5, с. 2083-2093
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  • 2015 Activity of 2-Aryl-2-(3-indolyl)acetohydroxamates against Drug-Resistant Cancer Cells
  • Aksenov Alexander V., Smirnov Alexander N., Magedov Igor V., Reisenauer Mary R., Aksenov Nicolai A., Aksenova Inna V., Pendleton Alexander L., Nguyen Gina, Johnston Robert K., Rubin Michael, De Carvalho Annelise, Kiss Robert, Mathieu Véronique, Lefranc Florence, Correa Jaime, Cavazos David A., Brenner Andrew J., Bryan Brad A., Rogelj Snezna, Kornienko Alexander, Frolova Liliya V.
  • в журнале Journal of Medicinal Chemistry, издательство American Chemical Society (United States), том 58, № 5, с. 2206-2220 DOI