European Journal of Medicinal Chemistryжурнал

Статьи, опубликованные в журнале

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• • The first series of 4,11-bis[(2-aminoethyl)amino]anthra[2,3-b]furan-5,10-diones: synthesis and anti-proliferative characteristics
  • Shchekotikhin A.E., Glazunova V.A., Dezhenkova L.G., Shevtsova E.K., Traven’ V.F., Balzarini J., H-S Huang, Shtil A.A., Preobrazhenskaya M.N.
  • в журнале European Journal of Medicinal Chemistry, издательство Elsevier BV (Netherlands), том 46, с. 213-218
• • 2023 C(21)-fluorinated thevinol scaffold for opioid ligands. 21,21,21-Trifluoro-6-O-nororvinols: Design, synthesis and analgesic activity
  • Sandulenko Irina V., Belozertseva Irina V., Zvartau Edwin E., Zelentsova Maria V., Ambartsumyan Asmik A., Smol'yakov Alexander F., Moiseev Sergey K.
  • в журнале European Journal of Medicinal Chemistry, издательство Elsevier BV (Netherlands), с. 115296 DOI
• • 2022 Discovery of the 4-aminopiperidine-based compound EM127 for the site-specific covalent inhibition of SMYD3
  • Parentia Marco Daniele, Naldi Marina, Manoni Elisabetta, Fabini Edoardo, Cederfelt Daniela, Talibove Vladimir O., Gressani Valeria, Guven Ummu, Grossi Valentina, Fasano Candida, Sanese Paola, De Marco Katia, Shtil Alexander A., Kurkin Alexander V., Altieri Andrea, Danielsone U.Helena, Caretti Giuseppina, Simone Cristiano, Varchi Greta, Bartolini Manuela, Del Rio Alberto
  • в журнале European Journal of Medicinal Chemistry, издательство Elsevier BV (Netherlands), с. 114683 DOI
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  • 2022 PSMA-targeted small-molecule docetaxel conjugate: Synthesis and preclinical evaluation
  • Machulkin A.E., Uspenskaya A.A., Zyk N.Y., Nimenko E.A., Ber A.P., Petrov S.A., Shafikov R.R., Skvortsov D.A., Smirnova G.B., Borisova Y.A., Pokrovsky V.S., Kolmogorov V.S., Vaneev A.N., Ivanenkov Y.A., Khudyakov A.D., Kovalev S.V., Erofeev A.S., Gorelkin P.V., Beloglazkina E.K., Zyk N.V., Khazanova E.S., Majouga A.G.
  • в журнале European Journal of Medicinal Chemistry, издательство Elsevier BV (Netherlands), том 227 DOI
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  • 2022 Synthesis, biological evaluation, and in silico studies of potential activators of apoptosis and carbonic anhydrase inhibitors on isatin-5-sulfonamide scaffold
  • Krymov Stepan K., Scherbakov Alexander M., Salnikova Diana I., Sorokin Danila V., Dezhenkova Lyubov G., Ivanov Ivan V., Vullo Daniela, De Luca Viviana, Capasso Clemente, Supuran Claudiu T., Shchekotikhin Andrey E.
  • в журнале European Journal of Medicinal Chemistry, издательство Elsevier BV (Netherlands), том 228 DOI
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  • 2021 Design of gp120 HIV-1 entry inhibitors by scaffold hopping via isosteric replacements
  • Iusupov Ildar R., Curreli Francesca, Spiridonov Evgeniy A., Markov Pavel O., Ahmed Shahad, Belov Dmitry S., Manasova Ekaterina V., Altieri Andrea, Kurkin Alexander V., Debnath Asim K.
  • в журнале European Journal of Medicinal Chemistry, издательство Elsevier BV (Netherlands), том 224 DOI
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  • 2021 Discovery of novel N4-alkylcytidines as promising antimicrobial agents
  • Alexandrova Liudmila A., Jasko Maxim V., Negrya Sergey D., Solyev Pavel N., Shevchenko Oleg V., Solodinin Andrei P., Kolonitskaya Daria P., Karpenko Inna L., Efremenkova Olga V., Glukhova Alla A., Boykova Yuliya V., Efimenko Tatiana A., Kost Natalya V., Avdanina Darya A., Nuraeva Gulgina K., Volkov Ivan A., Kochetkov Sergey N., Zhgun Alexander A.
  • в журнале European Journal of Medicinal Chemistry, издательство Elsevier BV (Netherlands) DOI
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  • 2021 Novel potent bifunctional carboxylesterase inhibitors based on a polyfluoroalkyl-2-imino-1,3-dione scaffold
  • Makhaeva G.F., Lushchekina S.V., Boltneva N.P., Serebryakova O.G., Kovaleva N.V., Rudakova E.V., Elkina N.A., Shchegolkov E.V., Burgart Y.V., Stupina T.S., Terentiev A.A., Radchenko E.V., Palyulin V.A., Saloutin V.I., Bachurin S.O., Richardson R.J.
  • в журнале European Journal of Medicinal Chemistry, издательство Elsevier BV (Netherlands), том 218, с. 113385 DOI
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  • 2021 PSMA-targeted low-molecular double conjugates for diagnostics and therapy
  • Petrov Stanislav A., Zyk Nikolay Y., Machulkin Aleksei E., Beloglazkina Elena K., Majouga Alexander G.
  • в журнале European Journal of Medicinal Chemistry, издательство Elsevier BV (Netherlands), том 225 DOI
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  • 2021 Phenoxazine nucleoside derivatives with a multiple activity against RNA and DNA viruses
  • Kozlovskaya Liubov I., Volok Viktor P., Shtro Anna A., Nikolaeva Yulia V., Chistov Alexey A., Matyugina Elena S., Belyaev Evgeny S., Jegorov Artjom V., Snoeck Robert, Korshun Vladimir A., Andrei Graciela, Osolodkin Dmitry I., Ishmukhametov Aydar A., Aralov Andrey V.
  • в журнале European Journal of Medicinal Chemistry, издательство Elsevier BV (Netherlands), том 220 DOI
• • 2021 Promising applications of steroid сonjugates for cancer research and treatment
  • Zolottsev V.A., Latysheva А.S., Pokrovsky V.S., Khan I.I., Misharin A.Y.
  • в журнале European Journal of Medicinal Chemistry, издательство Elsevier BV (Netherlands) DOI
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  • 2021 Thiophene-2-carboxamide derivatives of anthraquinone: A new potent antitumor chemotype
  • Volodina Yulia L., Tikhomirov Alexander S., Dezhenkova Lyubov G., Ramonova Alla A., Kononova Anastasia V., Andreeva Daria V., Kaluzhny Dmitry N., Schols Dominique, Moisenovich Mikhail M., Shchekotikhin Andrey E., Shtil Alexander A.
  • в журнале European Journal of Medicinal Chemistry, издательство Elsevier BV (Netherlands), том 221 DOI
• • 2020 6-Methyluracil derivatives as peripheral site ligand-hydroxamic acid conjugates: Reactivation for paraoxon-inhibited acetylcholinesterase
  • Semenov V.E., Zueva I.V., Lushchekina S.V., Lenina O.A., Gubaidullina L.M., Saifina L.F., Shulaeva M.M., Kayumova R.M., Saifina A.F., Gubaidullin A.T., Kondrashova S.A., Latypov S.K., Masson P., Petrov K.A.
  • в журнале European Journal of Medicinal Chemistry, издательство Elsevier BV (Netherlands), том 185 DOI
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  • 2020 Amides of Pyrrole- And Thiophene-Fused Anthraquinone Derivatives: A Role of the Heterocyclic Core in Antitumor Properties
  • Tikhomirov AS, Litvinova VA, Andreeva DV, Tsvetkov VB, Dezhenkova LG, Volodina YL, Kaluzhny DN, Treshalin ID, Schols D., Ramonova AA, Moisenovich MM, Shtil AA, Shchekotikhin AE
  • в журнале European Journal of Medicinal Chemistry, издательство Elsevier BV (Netherlands), том 199, с. 112294 DOI
• • 2020 Novel curcumin derivatives as P-glycoprotein inhibitors: Molecular modeling, synthesis and sensitization of multidrug resistant cells to doxorubicin
  • Sagnou Marina, Novikov Fedor N., Ivanova Ekaterina S., Alexiou Polyxeni, Stroylov Victor S., Titov Ilya Y., Tatarskiy Victor V., Vagida Murad S., Pelecanou Maria, Shtil Alexander A., Chilov Ghermes G.
  • в журнале European Journal of Medicinal Chemistry, издательство Elsevier BV (Netherlands) DOI
• • 2020 Phosphorus dendrimers as powerful nanoplatforms for drug delivery, as fluorescent probes and for liposome interaction studies: A concise overview
  • Shcharbin D., Bryszewska M., Mignani S., Shi X., Majoral J.P.
  • в журнале European Journal of Medicinal Chemistry, издательство Elsevier BV (Netherlands), том 208 DOI
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  • 2019 2-(2-(2,4-dioxopentan-3-ylidene)hydrazineyl)benzonitrile as novel inhibitor of receptor tyrosine kinase and PI3K/AKT/mTOR signaling pathway in glioblastoma
  • Anisha Viswanathan, Dinesh Kute, Aliyu Musa, Saravanan Konda Mani, ViliSipilä, Frank Emmert-Streib, Zubkov Fedor I., Gurbanov Atash V., Olli Yli-Harja, Meenakshisundaram Kandhavelu
  • в журнале European Journal of Medicinal Chemistry, издательство Elsevier BV (Netherlands), том 166, с. 291-303 DOI
• • 2019 Chikungunya virus inhibition by synthetic Coumarin-Guanosine conjugates
  • Hwu Jih Ru, Huang Wen-Chieh, Lin Shu-Yu, Tan Kui-Thong, Yu-Chen Hu, Shieh Fa-Kuen, Bachurin Sergey O., Ustyugov Aleksey, Tsay Shwu-Chen
  • в журнале European Journal of Medicinal Chemistry, издательство Elsevier BV (Netherlands) DOI
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  • 2019 Compounds based on 5-(perylen-3-ylethynyl)uracil scaffold: High activity against tick-borne encephalitis virus and non-specific activity against enterovirus A
  • Chistov Alexey A., Orlov Alexey A., Streshnev Philipp P., Slesarchuk Nikita A., Aparin Ilya O., Brijesh Rathi, Brylev Vladimir A., Kutyakov Sergey V., Mikhura Irina V., Ustinov Alexey V., Gunnar Westman, Palyulin Vladimir A., Nidhi Jain, Osolodkin Dmitry I., Kozlovskaya Liubov I., Korshun Vladimir A.
  • в журнале European Journal of Medicinal Chemistry, издательство Elsevier BV (Netherlands), том 171, с. 93-103 DOI
• • 2019 Investigating 1,2,3,4,5,6-hexahydroazepino[4,3-b]indole as scaffold of butyrylcholinesterase-selective inhibitors with additional neuroprotective activities for Alzheimer's disease
  • Purgatorio R., Catto M.de Candia; M, Carrieri A., Pisani L., De Palma A., Toma M., Ivanova O.A., Voskressensky L.G., Altomare C.D.
  • в журнале European Journal of Medicinal Chemistry, издательство Elsevier BV (Netherlands) DOI
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  • 2019 New 2,6-diaminopyridines containing a sterically hindered benzylphosphonate moiety in the aromatic core as potential antioxidant and anti-cancer drugs
  • Gibadullina Elmira, Nguyen Thi Thu, Strelnik Anna, Sapunova Anastasiia, Voloshina Alexandra, Sudakov Igor, Vyshtakalyuk Alexandra, Voronina Julya, Pudovik Michael, Burilov Alexander
  • в журнале European Journal of Medicinal Chemistry, издательство Elsevier BV (Netherlands), том 184, с. 111735 DOI
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  • 2019 New anthra[2,3-b]furancarboxamides: A role of positioning of the carboxamide moiety in antitumor properties
  • Volodina Y.L., Dezhenkova L.G., Tikhomirov A.S., Tatarskiy V.V., Kaluzhny D.N., Moisenovich A.M., Moisenovich M.M., Isagulieva A.K., Shtil A.A., Tsvetkov V.B., Shchekotikhin A.E.
  • в журнале European Journal of Medicinal Chemistry, издательство Elsevier BV (Netherlands), том 165, с. 31-45 DOI
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  • 2019 New anthra[2,3-b]furancarboxamides: A role of positioning of the carboxamide moiety in antitumor properties
  • Volodina YL, Dezhenkova LG, Tikhomirov AS, Tatarskiy VV, Kaluzhny DN, Moisenovich AM, Moisenovich MM, Isagulieva AK, Shtil AA, Tsvetkov VB, Shchekotikhin AE
  • в журнале European Journal of Medicinal Chemistry, издательство Elsevier BV (Netherlands), № 165, с. 31-45 DOI
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  • 2019 Novel tyrosyl-DNA phosphodiesterase 1 inhibitors enhance the therapeutic impact of topotecan on in vivo tumor models
  • Zakharenko A.L., Luzina O.A., Sokolov D.N., Kaledin V.I., Nikolin V.P., Popova N.A., Patel J., Zakharova O.D., Chepanova A.A., Zafar A., Reynisson J., Leung E., Leung I.K.H, Volcho K.P., Salakhutdinov N.F., Lavrik O.I.
  • в журнале European Journal of Medicinal Chemistry, издательство Elsevier BV (Netherlands), том 161, с. 581-593 DOI
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  • 2019 Steroidal N-Sulfonylimidates: Synthesis and biological evaluation in breast cancer cells
  • Volkova Yulia A., Kozlov Andrey S., Kolokolova Marya K., Uvarov Denis Y., Gorbatov Sergey A., Andreeva Olga E., Scherbakov Alexander M., Zavarzin Igor V.
  • в журнале European Journal of Medicinal Chemistry, издательство Elsevier BV (Netherlands), том 179, с. 694-706 DOI